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Official PDF TranslationActa Biochimica et Biophysica Sinica

Withaferin A combined with ricolinostat: a potent synergistic therapy for cervical cancer through regulating p53 ubiquitination and acetylation

Authors: CHEN Tian; XU Yiting; YANG Kunming; DU Yutong; ZHU Zhuan; XU Lingling; WANG Xinrong; YIN Yi; HU Yu; WANG Chengcheng; HU Ronggui; LI Chuanyin

DOI: 10.3724/abbs.2025048Status: Verified Translated Edition
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Key Findings in This Report

• • Combination of WA and RIC yields a combination index (CI) < 1 in HeLa, SiHa, and Caski cells, indicating synergistic inhibition of cell viability; this synergy is critical for reducing effective doses and minimizing off-target toxicity in clinical settings. • • WA treatment for 24 h disrupts the p53-E6AP interaction, decreasing p53 ubiquitination; this directly addresses the primary degradation pathway in HPV-positive cervical cancer, potentially restoring p53 tumor-suppressive function. • • RIC treatment for 24 h inhibits HDAC6-mediated deacetylation, increasing p53 acetylation; elevated acetylation enhances p53 stability and transcriptional activity, a mechanism that complements ubiquitination blockade. • • The combination extends p53 half-life beyond 60 min in cycloheximide chase assays, compared to rapid degradation in controls; this sustained stabilization is essential for mounting an effective apoptotic response and overcoming the short half-life bottleneck of wild-type p53 in cervical cancer.